BDBM50121900 Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pro-Val-NH2::CHEMBL439490
SMILES CCCC[C@H](NC(=O)C(CO)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CO)NC(C)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@H](Cc1ccccc1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCC(=O)N[C@@H](CCCCN)C(=O)N1CCC[C@@H]1C(=O)N[C@H](C(C)C)C(N)=O
InChI Key InChIKey=UAHFGYDRQSXQEB-BVMGHOOCSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 13 hits for monomerid = 50121900
TargetMelanocortin receptor 5(Homo sapiens (Human))
H. Lee Moffitt Cancer Center & Research Institute
Curated by ChEMBL
H. Lee Moffitt Cancer Center & Research Institute
Curated by ChEMBL
Affinity DataKi: 9.90nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC5 receptor expressed in human HEK293 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0860nMAssay Description:Functional activity at the mouse melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0710nMAssay Description:In vitro activaction of mouse recombinant Melanocortin-5 receptor.More data for this Ligand-Target Pair
Affinity DataEC50: 0.0710nMAssay Description:Activity in mouse melanocortin-5 receptor stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0710nMAssay Description:Agonist activity towards mouse Melanocortin-5 receptor (mMC5R)More data for this Ligand-Target Pair
Affinity DataEC50: 0.0710nMAssay Description:Effective concentration against mouse Melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0950nMAssay Description:Effective concentration for mouse Melanocortin-5 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0780nMAssay Description:In vitro agonist potency for Mouse Melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0620nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.280nMAssay Description:Agonist activity at mouse MC5 receptor expressed in HEK293 cells after 6 hrs by cAMP-based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.170nMAssay Description:Agonistic activity against mouse MC5RMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0780nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.260nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair